SCHEMBL8312296

SCHEMBL8312296

CS(=O)(=O)N1CC[C@@](OCc2ccccc2)(c2ccc(Cl)cc2)[C@H](OCc2ccc(F)c(F)c2F)C1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
TACR1 P25103 1/20 0.33
CCR1 P32246 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
RORC P51449 1/20 0.32
TP53 P04637 1/20 0.31
MDM2 Q00987 1/20 0.31
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
POLB P06746 1/20 0.31
TSHR P16473 2/20 0.31
CYP3A4 P08684 1/20 0.31
PGR P06401 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP1A2 P05177 1/20 0.30
HIF1A Q16665 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6095667 0.85 CCR1 (0.39) CYP2D6MEN1KMT2ACCR1ALDH1A1
SCHEMBL6095673 0.85 CCR1 (0.39) CYP2D6MEN1KMT2ACCR1ALDH1A1
SCHEMBL6274732 0.84 CCR3 (0.34) CCR1ALDH1A1
SCHEMBL6095902 0.83 CCR1 (0.38) CCR1OPRD1OPRK1ALDH1A1SMN1; SMN2
SCHEMBL6095898 0.83 CCR1 (0.38) CCR1OPRD1OPRK1ALDH1A1SMN1; SMN2
SCHEMBL6841776 0.82 BCHE (0.33) CCR1
SCHEMBL6098489 0.79 DRD4 (0.36) CCR1ALDH1A1
SCHEMBL6098492 0.79 DRD4 (0.36) CCR1ALDH1A1
SCHEMBL8306421 0.79 DRD4 (0.36) CCR1ALDH1A1
SCHEMBL8307328 0.78 SLC6A2 (0.36) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080460-A1 SUBSTITUTED PIPERIDINES AS NOVEL MDM2-p53 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2004-09-23 WO disclosed