SCHEMBL8312622

SCHEMBL8312622

Oc1ccc2oc(-c3nc(-c4ccccc4)cs3)cc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.51
MAPT P10636 3/20 0.51
MEN1 O00255 2/20 0.51
ALDH1A1 P00352 2/20 0.51
HPGD P15428 2/20 0.51
MAPK1 P28482 2/20 0.51
NPSR1 Q6W5P4 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
ESR1 P03372 1/20 0.50
ESR2 Q92731 1/20 0.50
HSD17B1 P14061 1/20 0.50
HSD17B2 P37059 1/20 0.50
CYP19A1 P11511 3/20 0.47
KDM4E B2RXH2 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47
ALOX12 P18054 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311831 0.84 MAPT (0.63) KMT2AMAPTMEN1ALDH1A1MAPK1
SCHEMBL8311567 0.84 CYP19A1 (0.53) KMT2AMAPTMEN1ALDH1A1MAPK1
SCHEMBL5940765 0.84 MIF (0.67) KMT2AMAPTMEN1ALDH1A1HPGD
SCHEMBL8314667 0.82 MEN1 (0.52) KMT2AMAPTMEN1ALDH1A1HPGD
SCHEMBL8312888 0.81 MAPT (0.56) KMT2AMAPTMEN1ALDH1A1HPGD
SCHEMBL7328614 0.78 ESR1 (0.79) MAPTESR1ESR2HSD17B1CYP19A1
SCHEMBL8310912 0.78 MIF (0.54) MAPTALDH1A1HPGDESR1ESR2
SCHEMBL8311480 0.76 ESR1 (0.47) MAPTESR1ESR2CYP19A1MIF
SCHEMBL8315191 0.76 MAPK1 (0.41) KMT2AMAPTMEN1ALDH1A1HPGD
SCHEMBL6600736 0.75 ESR1 (0.48) KMT2AMEN1ALDH1A1HPGDESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528337-B1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1999-10-20 EP disclosed
CN-1033088-C Thiazolylbenzofuran derivatives, processes for preparation thereof and pharmaceutical composition comprising same FUJISAWA PHARMACEUTICAL CO (JP) 1996-10-23 CN disclosed
US-5296495-A Antiallergens, antiinflammatory FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-03-22 US disclosed
EP-0528337-A1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-02-24 EP disclosed