SCHEMBL8311567

SCHEMBL8311567

Oc1ccc2oc(-c3nc(-c4ccccn4)cs3)cc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.53
MBD2 Q9UBB5 1/20 0.46
NR4A1 P22736 1/20 0.46
VCP P55072 1/20 0.46
KDM4E B2RXH2 3/20 0.46
MAPT P10636 2/20 0.46
ALDH1A1 P00352 2/20 0.46
RAB9A P51151 2/20 0.46
PKM P14618 1/20 0.46
GFER P55789 1/20 0.46
HSD17B10 Q99714 1/20 0.46
KDM4C Q9H3R0 1/20 0.46
PDE4D Q08499 3/20 0.46
GRIA1 P42261 1/20 0.44
MEN1 O00255 1/20 0.44
HSP90AA1 P07900 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312622 0.84 KMT2A (0.51) CYP19A1VCPKDM4EMAPTALDH1A1
SCHEMBL8310447 0.82 CYP19A1 (0.50) CYP19A1KDM4EMAPTALDH1A1RAB9A
SCHEMBL8314667 0.79 MEN1 (0.52) CYP19A1VCPKDM4EMAPTALDH1A1
SCHEMBL8315476 0.78 CYP19A1 (0.43) CYP19A1KDM4EMAPTALDH1A1RAB9A
SCHEMBL8314218 0.76 CYP19A1 (0.41) CYP19A1KDM4EMAPTALDH1A1RAB9A
SCHEMBL8310912 0.75 MIF (0.54) KDM4EMAPTALDH1A1RAB9AHSD17B10
SCHEMBL8311831 0.74 MAPT (0.63) CYP19A1VCPKDM4EMAPTALDH1A1
SCHEMBL8311480 0.73 ESR1 (0.47) CYP19A1MAPTRAB9APDE4DMIF
SCHEMBL8311144 0.72 ESR1 (0.48) KDM4EALDH1A1HSD17B10PDE4DSMN1; SMN2
SCHEMBL8312572 0.72 ESR1 (0.48) KDM4EALDH1A1HSD17B10PDE4DSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528337-B1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1999-10-20 EP disclosed
CN-1036589-C New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1997-12-03 CN disclosed
CN-1033088-C Thiazolylbenzofuran derivatives, processes for preparation thereof and pharmaceutical composition comprising same FUJISAWA PHARMACEUTICAL CO (JP) 1996-10-23 CN disclosed
US-5296495-A Antiallergens, antiinflammatory FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-03-22 US disclosed
EP-0528337-A1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-02-24 EP disclosed