SCHEMBL8313247

SCHEMBL8313247

CC(C)(C)OC(=O)N1[C@H](C(=O)Cl)C[C@@H]2CCCC[C@@H]21

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.49
CHRM3 P20309 1/20 0.49
PREP P48147 5/20 0.42
EPHX1 P07099 1/20 0.37
HSD11B1 P28845 1/20 0.36
NR1H2 P55055 2/20 0.36
HPGD P15428 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.35
GPR119 Q8TDV5 1/20 0.35
ACE P12821 1/20 0.34
NR1H3 Q13133 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4847115 0.88 CHRM2 (0.45) CHRM2CHRM1CHRM3PREPEPHX1
SCHEMBL3050914 0.88 CHRM2 (0.45) CHRM2CHRM1CHRM3PREPEPHX1
SCHEMBL4840543 0.88 CHRM2 (0.45) CHRM2CHRM1CHRM3PREPEPHX1
SCHEMBL8337646 0.88 CHRM2 (0.45) CHRM2CHRM1CHRM3PREPEPHX1
SCHEMBL14053968 0.88 CHRM2 (0.45) CHRM2CHRM1CHRM3PREPEPHX1
SCHEMBL4795338 0.88 CHRM2 (0.45) CHRM2CHRM1CHRM3PREPEPHX1
SCHEMBL15116700 0.88 CHRM2 (0.45) CHRM2CHRM1CHRM3PREPEPHX1
SCHEMBL20221211 0.88 CHRM2 (0.45) CHRM2CHRM1CHRM3PREPEPHX1
SCHEMBL1336739 0.88 CHRM2 (0.45) CHRM2CHRM1CHRM3PREPEPHX1
SCHEMBL27272431 0.88 CHRM2 (0.45) CHRM2CHRM1CHRM3PREPEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004071454-A2 SUBSTITUTED AZETIDINE COMPOUNDS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE IV GUILFORD PHARMACEUTICALS INC. (US) 2004-08-26 WO disclosed