SCHEMBL8313626

SCHEMBL8313626

O=[N+]([O-])c1cccc(Nc2ncnc3cnc(NC4CCC(O)CC4)nc23)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.56
GSK3B P49841 1/20 0.56
FLT3 P36888 1/20 0.55
TYRO3 Q06418 1/20 0.55
MERTK Q12866 1/20 0.55
GAS6 Q14393 1/20 0.55
BRAF P15056 1/20 0.53
ABCG2 Q9UNQ0 2/20 0.50
EGFR P00533 9/20 0.48
ERBB2 P04626 1/20 0.47
HPGD P15428 1/20 0.47
HTT P42858 1/20 0.47
MAPK8 P45983 1/20 0.46
MAPK9 P45984 1/20 0.46
CTSL P07711 2/20 0.45
CTSB P07858 2/20 0.45
CTSS P25774 2/20 0.45
CTSK P43235 2/20 0.45
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313619 1.00 GSK3A (0.56) GSK3AGSK3BFLT3TYRO3MERTK
SCHEMBL8313945 1.00 GSK3A (0.56) GSK3AGSK3BFLT3TYRO3MERTK
SCHEMBL8315091 0.95 ABCG2 (0.54) GSK3AGSK3BFLT3TYRO3MERTK
SCHEMBL8317920 0.91 EGFR (0.51) GSK3AGSK3BFLT3TYRO3MERTK
SCHEMBL8317918 0.91 EGFR (0.51) GSK3AGSK3BFLT3TYRO3MERTK
SCHEMBL8315283 0.90 ABCG2 (0.48) GSK3AGSK3BFLT3TYRO3MERTK
SCHEMBL8315275 0.90 ABCG2 (0.48) GSK3AGSK3BFLT3TYRO3MERTK
SCHEMBL8315077 0.90 FLT3 (0.47) GSK3AGSK3BFLT3TYRO3MERTK
SCHEMBL8315087 0.90 FLT3 (0.47) GSK3AGSK3BFLT3TYRO3MERTK
SCHEMBL8316755 0.89 CTSL (0.57) GSK3AGSK3BFLT3TYRO3MERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed