SCHEMBL8313749

SCHEMBL8313749

Cc1ccc(C[C@H]2CCN(Cc3nc4ccc(O)cc4[nH]3)C[C@@H]2O)cc1

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 10/20 0.74
GRIN2B Q13224 10/20 0.74
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5235290 0.92 GRIN1 (0.62) GRIN1GRIN2BALDH1A1GAA
SCHEMBL5235300 0.92 GRIN1 (0.62) GRIN1GRIN2BALDH1A1GAA
SCHEMBL5235309 0.92 GRIN1 (0.62) GRIN1GRIN2BALDH1A1GAA
SCHEMBL8318042 0.85 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL6001498 0.82 GRIN2B (0.61) GRIN1GRIN2BGAAPKMTSHR
SCHEMBL6001504 0.82 GRIN2B (0.61) GRIN1GRIN2BGAAPKMTSHR
SCHEMBL6001501 0.82 GRIN2B (0.61) GRIN1GRIN2BGAAPKMTSHR
SCHEMBL5269544 0.77 GRIN1 (0.84) GRIN1GRIN2B
SCHEMBL8313704 0.75 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8313723 0.74 GRIN1 (1.00) GRIN1GRIN2BGAAPKMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048364-A1 2-[(4-BENZYL)-1-PIPERIDINYL)METHYL]BENZIMIDAZOLE-5-OL DERIVATIVES AS NR2B RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2004-06-10 WO disclosed