SCHEMBL8313723

SCHEMBL8313723

Oc1ccc2nc(CN3CCC(Cc4ccccc4)CC3)[nH]c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 11/20 1.00
GRIN2B Q13224 11/20 1.00
GAA P10253 1/20 0.57
PKM P14618 1/20 0.57
TSHR P16473 1/20 0.57
THRB P10828 1/20 0.55
GRIN2D O15399 1/20 0.53
GRIN3B O60391 1/20 0.53
GRIN2A Q12879 1/20 0.53
GRIN2C Q14957 1/20 0.53
GRIN3A Q8TCU5 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5237195 0.91 GRIN1 (0.84) GRIN1GRIN2BGAATHRBGRIN2D
SCHEMBL8313704 0.89 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8318042 0.89 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8320273 0.89 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8312848 0.86 GRIN1 (0.80) GRIN1GRIN2B
SCHEMBL1388535 0.86 GRIN2B (1.00) GRIN1GRIN2BTHRBGRIN2AGRIN2C
SCHEMBL8318192 0.85 GRIN1 (1.00) GRIN1GRIN2BGAA
SCHEMBL8319076 0.84 GRIN1 (1.00) GRIN1GRIN2BGAA
SCHEMBL8313716 0.81 GRIN1 (0.67) GRIN1GRIN2BGAAPKMTSHR
SCHEMBL5269544 0.81 GRIN1 (0.84) GRIN1GRIN2BTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048364-A1 2-[(4-BENZYL)-1-PIPERIDINYL)METHYL]BENZIMIDAZOLE-5-OL DERIVATIVES AS NR2B RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2004-06-10 WO disclosed