SCHEMBL8314012

SCHEMBL8314012

FC(F)(F)Oc1cccc(Nc2ncnc3cnc(NC4CC4)nc23)c1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SYK P43405 2/20 0.53
EGFR P00533 5/20 0.52
ERBB2 P04626 1/20 0.52
HPGD P15428 1/20 0.52
HTT P42858 1/20 0.52
CTSC P53634 2/20 0.49
GALR2 O43603 1/20 0.48
GALR1 P47211 1/20 0.48
CTSL P07711 1/20 0.48
CTSB P07858 1/20 0.48
CTSS P25774 1/20 0.48
CTSK P43235 1/20 0.48
BRAF P15056 5/20 0.47
CSNK2A1 P68400 2/20 0.47
PIM1 P11309 2/20 0.45
CSNK2A2 P19784 1/20 0.45
CSNK2B P67870 1/20 0.45
CSNK2A3 Q8NEV1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998709 0.95 BRAF (0.50) SYKEGFRERBB2HPGDHTT
SCHEMBL6998715 0.95 BRAF (0.50) SYKEGFRERBB2HPGDHTT
SCHEMBL6993308 0.88 BRAF (0.48) SYKEGFRERBB2HPGDHTT
SCHEMBL6993311 0.88 BRAF (0.48) SYKEGFRERBB2HPGDHTT
SCHEMBL8312571 0.87 CSNK2A1 (0.60) SYKEGFRERBB2HPGDHTT
SCHEMBL8317346 0.85 EGFR (0.51) EGFRERBB2HPGDHTTCTSC
SCHEMBL8318987 0.85 CTSC (0.61) EGFRERBB2HPGDHTTCTSC
SCHEMBL8317921 0.84 BRAF (0.52) EGFRERBB2HPGDHTTGALR2
SCHEMBL8317917 0.84 BRAF (0.52) EGFRERBB2HPGDHTTGALR2
SCHEMBL8317928 0.83 EGFR (0.60) EGFRERBB2HPGDHTTBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed