SCHEMBL8314038

SCHEMBL8314038

CN(C(=O)C(F)(F)F)[C@](CSCc1ccccc1)(CC(Cl)(Cl)Cl)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.35
CES1 P23141 6/20 0.35
HDAC4 P56524 5/20 0.35
HDAC6 Q9UBN7 5/20 0.35
HDAC3 O15379 2/20 0.35
HDAC1 Q13547 2/20 0.35
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
MLYCD O95822 1/20 0.33
FAAH O00519 3/20 0.33
RIPK1 Q13546 1/20 0.32
LIPE Q05469 1/20 0.32
TP53 P04637 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311399 0.68 PPARA (0.37) CYP2C19CES1PPARGPPARA
SCHEMBL8314036 0.68 PPARA (0.36) CYP2C19CES1HDAC4HDAC6HDAC3
SCHEMBL8232709 0.67 PPARA (0.47) CYP2C19PPARGPPARA
SCHEMBL8922764 0.67 PPARG (0.42) CYP2C19CES1HDAC4HDAC6HDAC3
SCHEMBL1713309 0.67 CES1 (0.44) CYP2C19CES1POLB
SCHEMBL9171687 0.66 CYP2C19 (0.50) CYP2C19PPARGPPARARIPK1
SCHEMBL4103416 0.65 PPARG (0.40) CYP2C19CES1PPARGPPARARIPK1
SCHEMBL4103411 0.65 PPARG (0.40) CYP2C19CES1PPARGPPARARIPK1
SCHEMBL9301235 0.64 CYP2C19 (0.47) CYP2C19PPARGPPARARIPK1
SCHEMBL4099299 0.64 CYP2C19 (0.47) CYP2C19PPARGPPARAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724601-A4 S 3N CHELATING COMPOUNDS FOR THE RADIOLABELING OF LIGANDS, ANTI-LIGANDS OR OTHER PROTEINS NEORX CORP (US) 1999-02-03 EP disclosed
US-5684137-A TECHNETIUM AND RHENIUM LABELS FOR LIGANDS AND PROTEINS NEORX CORPORATION (US) 1997-11-04 US disclosed
EP-0724601-A1 S 3N CHELATING COMPOUNDS FOR THE RADIOLABELING OF LIGANDS, ANTI-LIGANDS OR OTHER PROTEINS NEORX CORPORATION (US) 1996-08-07 EP disclosed
WO-1995005398-A1 S3N CHELATING COMPOUNDS FOR THE RADIOLABELING OF LIGANDS, ANTI-LIGANDS OR OTHER PROTEINS NEORX CORPORATION (US) 1995-02-23 WO disclosed