SCHEMBL8311399

SCHEMBL8311399

O=C(O)[C@H](CSCc1ccccc1)N(CC(Cl)(Cl)Cl)C(=O)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 6/20 0.37
PPARG P37231 4/20 0.37
ACE P12821 1/20 0.36
CYP2C19 P33261 1/20 0.35
CES1 P23141 2/20 0.35
CPA1 P15085 1/20 0.35
PPARD Q03181 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4462979 0.85 PPARG (0.40) PPARAPPARGACECYP2C19CES1
SCHEMBL8310840 0.82 PPARA (0.42) PPARAPPARGACECYP2C19PPARD
SCHEMBL8922764 0.82 PPARG (0.42) PPARAPPARGACECYP2C19CES1
SCHEMBL8314036 0.77 PPARA (0.36) PPARAPPARGACECYP2C19CES1
SCHEMBL8310839 0.70 ACE (0.42) PPARAPPARGACECYP2C19
SCHEMBL18270379 0.68 PPARA (0.47) PPARAPPARGACECYP2C19
SCHEMBL4983034 0.68 PPARA (0.47) PPARAPPARGACECYP2C19
SCHEMBL8314038 0.68 CYP2C19 (0.35) PPARAPPARGCYP2C19CES1
SCHEMBL10420286 0.68 MEN1 (0.43) CYP2C19CES1CPA1
SCHEMBL10420288 0.68 MEN1 (0.43) CYP2C19CES1CPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724601-A4 S 3N CHELATING COMPOUNDS FOR THE RADIOLABELING OF LIGANDS, ANTI-LIGANDS OR OTHER PROTEINS NEORX CORP (US) 1999-02-03 EP disclosed
US-5684137-A TECHNETIUM AND RHENIUM LABELS FOR LIGANDS AND PROTEINS NEORX CORPORATION (US) 1997-11-04 US disclosed
EP-0724601-A1 S 3N CHELATING COMPOUNDS FOR THE RADIOLABELING OF LIGANDS, ANTI-LIGANDS OR OTHER PROTEINS NEORX CORPORATION (US) 1996-08-07 EP disclosed
WO-1995005398-A1 S3N CHELATING COMPOUNDS FOR THE RADIOLABELING OF LIGANDS, ANTI-LIGANDS OR OTHER PROTEINS NEORX CORPORATION (US) 1995-02-23 WO disclosed