SCHEMBL8314464

SCHEMBL8314464

CN(C)C1CCC(Nc2ncc3ncnc(Nc4ccc(Cl)c(Cl)c4)c3n2)CC1

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.63
ERBB2 P04626 1/20 0.63
HPGD P15428 1/20 0.63
HTT P42858 1/20 0.63
IRAK4 Q9NWZ3 18/20 0.52
BRAF P15056 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314462 1.00 EGFR (0.63) EGFRERBB2HPGDHTTIRAK4
SCHEMBL8316240 0.92 EGFR (0.69) EGFRERBB2HPGDHTTBRAF
SCHEMBL6989676 0.92 EGFR (0.76) EGFRERBB2HPGDHTTIRAK4
SCHEMBL3473824 0.92 EGFR (0.76) EGFRERBB2HPGDHTTIRAK4
SCHEMBL8316363 0.88 EGFR (0.57) EGFRERBB2HPGDHTTIRAK4
SCHEMBL8316360 0.88 EGFR (0.57) EGFRERBB2HPGDHTTIRAK4
SCHEMBL8315348 0.87 EGFR (0.64) EGFRERBB2HPGDHTTBRAF
SCHEMBL8313702 0.87 EGFR (0.64) EGFRERBB2HPGDHTTIRAK4
SCHEMBL8313697 0.87 EGFR (0.64) EGFRERBB2HPGDHTTIRAK4
SCHEMBL8315620 0.87 EGFR (0.64) EGFRERBB2HPGDHTTBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed