SCHEMBL8316240

SCHEMBL8316240

Clc1ccc(Nc2ncnc3cnc(NC4CC4)nc23)cc1Cl

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.69
ERBB2 P04626 4/20 0.69
HPGD P15428 1/20 0.69
HTT P42858 1/20 0.69
CSNK2A1 P68400 2/20 0.48
BRAF P15056 2/20 0.48
BCL6 P41182 2/20 0.45
MAPT P10636 1/20 0.45
EPHA2 P29317 3/20 0.43
KDR P35968 3/20 0.43
EPHB4 P54760 3/20 0.43
CSNK2A2 P19784 1/20 0.43
CSNK2B P67870 1/20 0.43
CTSC P53634 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315620 0.95 EGFR (0.64) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8313697 0.95 EGFR (0.64) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8315348 0.95 EGFR (0.64) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8313702 0.95 EGFR (0.64) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8315344 0.95 EGFR (0.64) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8318062 0.93 EGFR (0.64) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8314200 0.93 EGFR (0.64) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8316366 0.92 EGFR (0.63) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8314464 0.92 EGFR (0.63) EGFRERBB2HPGDHTTBRAF
SCHEMBL8316373 0.92 EGFR (0.63) EGFRERBB2HPGDHTTCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP claimed
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
US-5707989-A ANTITUMOR AGENTS, INHIBITING SIGNAL TRANSDUCTION MEDIATED BY TYROSINE KINASES DR. KARL THOMAE GMBH (DE) 1998-01-13 US disclosed