SCHEMBL8314795

SCHEMBL8314795

Fc1ccc(Nc2ncnc3cnc(-c4ccccc4)nc23)cc1Cl

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 0.59
ABCG2 Q9UNQ0 1/20 0.58
ERBB2 P04626 7/20 0.55
HPGD P15428 1/20 0.55
HTT P42858 1/20 0.55
GRM1 Q13255 1/20 0.55
MAPT P10636 1/20 0.51
CD38 P28907 1/20 0.48
FBP1 P09467 2/20 0.48
AURKA O14965 1/20 0.48
INSR P06213 1/20 0.48
PDGFRB P09619 1/20 0.48
FLT4 P35916 1/20 0.48
KDR P35968 1/20 0.48
CLK1 P49759 1/20 0.48
EPHB4 P54760 1/20 0.48
TEK Q02763 1/20 0.48
AURKB Q96GD4 1/20 0.48
ERBB4 Q15303 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8317382 0.86 EGFR (0.54) EGFRERBB2HPGDHTTGRM1
SCHEMBL6992452 0.81 GRM1 (0.65) EGFRERBB2HPGDHTTGRM1
SCHEMBL8319146 0.81 EGFR (0.61) EGFRERBB2HPGDHTTGRM1
SCHEMBL8319823 0.79 EGFR (0.64) EGFRERBB2HPGDHTTGRM1
SCHEMBL6994181 0.79 EGFR (0.58) EGFRERBB2HPGDHTTGRM1
SCHEMBL8314618 0.78 EGFR (0.61) EGFRERBB2HPGDHTTGRM1
SCHEMBL8484377 0.78 EGFR (0.64) EGFRERBB2HPGDHTTGRM1
SCHEMBL30127056 0.77 EGFR (0.63) EGFRERBB2HPGDHTTGRM1
SCHEMBL7000275 0.77 EGFR (0.64) EGFRERBB2HPGDHTTGRM1
SCHEMBL6993701 0.77 EGFR (0.64) EGFRERBB2HPGDHTTGRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed