SCHEMBL8314975

SCHEMBL8314975

O=C1c2cc3c(cc2OC2CCCN12)C(=O)N1CCCC1O3

nearest known ligand 0.82

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.82
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
GAA P10253 1/20 0.33
CDK4 P11802 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
MAPT P10636 1/20 0.30
ALOX15 P16050 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8367567 0.95 GRIA1 (0.75) GRIA1ALDH1A1HPGDHSD17B10GAA
SCHEMBL8367555 0.95 GRIA1 (0.80) GRIA1ALDH1A1HPGDHSD17B10GAA
SCHEMBL12049626 0.91 GRIA1 (0.84) GRIA1ALDH1A1KDM4EMAPTKMT2A
SCHEMBL29542563 0.91 GRIA1 (1.00) GRIA1HPGDMEN1KMT2A
SCHEMBL678000 0.91 GRIA1 (1.00) GRIA1HPGDMEN1KMT2A
SCHEMBL31562972 0.91 GRIA1 (0.84) GRIA1ALDH1A1KDM4EMAPTKMT2A
SCHEMBL8368751 0.88 GRIA1 (0.71) GRIA1
SCHEMBL8368729 0.87 GRIA1 (0.69) GRIA1ALDH1A1HPGDHSD17B10GAA
SCHEMBL8366785 0.87 GRIA1 (0.69) GRIA1
SCHEMBL8367564 0.87 GRIA1 (0.69) GRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7799913-B2 Carbonylbenzoxazine compounds for enhancing glutamatergic synaptic responses CORTEX PHARMACEUTICALS, INC. (US) 2010-09-21 US disclosed
US-7799913-B2 Carbonylbenzoxazine compounds for enhancing glutamatergic synaptic responses CORTEX PHARMACEUTICALS, INC. (US) 2010-09-21 US disclosed
WO-2004062616-A2 METHOD OF TREATING COGNITIVE DECLINE DUE TO SLEEP DEPRIVATION AND STRESS CORTEX PHARMACEUTICALS, INC. (US) 2004-07-29 WO disclosed
WO-2003045315-A2 CARBONYLBENZOXAZINE COMPOUNDS FOR ENHANCING GLUTAMATERGIC SYNAPTIC RESPONSES CORTEX PHARMACEUTICALS, INC. (US) 2003-06-05 WO disclosed