SCHEMBL8315451

SCHEMBL8315451

CCOC(=O)OC1CNCCN1C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.41
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
ALDH1A1 P00352 3/20 0.34
TSHR P16473 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NR1H3 Q13133 2/20 0.31
NR1H2 P55055 1/20 0.31
ADORA1 P30542 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043813 0.84 PARP1 (0.44) PARP1MEN1KMT2AALDH1A1NR1H2
SCHEMBL29289211 0.84 PARP1 (0.44) PARP1MEN1KMT2AALDH1A1NR1H2
SCHEMBL27722775 0.82 PARP1 (0.45) PARP1HSD17B10KDM4EMAPTTHRB
SCHEMBL27717164 0.82 PARP1 (0.45) PARP1HSD17B10KDM4EMAPTTHRB
SCHEMBL18789978 0.80 PARP1 (0.41) PARP1ALDH1A1HSD17B10
SCHEMBL28135174 0.79 PARP1 (0.44) PARP1HSD17B10KDM4EMAPTTHRB
SCHEMBL28094553 0.79 PARP1 (0.44) PARP1HSD17B10KDM4EMAPTTHRB
SCHEMBL6541621 0.79 PARP1 (0.43) PARP1MEN1KMT2AALDH1A1TSHR
SCHEMBL7054243 0.79 PARP1 (0.43) PARP1MEN1KMT2AALDH1A1TSHR
SCHEMBL7056396 0.79 PARP1 (0.43) PARP1MEN1KMT2AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623615-B1 Substituted 1-phenyl-oxazolidin-2-one derivatives, their preparation and their use as adhesion-receptor antagonists MERCK PATENT GMBH (DE) 1999-06-30 EP disclosed
EP-0623615-A1 Adhesion-receptor antagonists MERCK PATENT GmbH (DE) 1994-11-09 EP disclosed