SCHEMBL8315663

SCHEMBL8315663

O=CNC1c2ccc(Cl)cc2-c2[nH]c(=O)c3nccn3c21

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIA1 P42261 1/20 0.39
GRIA2 P42262 1/20 0.39
GRIA3 P42263 1/20 0.39
GRIA4 P48058 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1387922 0.88 GRIN2D (0.40) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL7847268 0.85 GRIN2D (0.38) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL1387540 0.84 PDE2A (0.42)
SCHEMBL1388118 0.83 GRIN2D (0.41) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL1388184 0.80 CCKBR (0.40)
SCHEMBL1387825 0.77
SCHEMBL1387813 0.71 PDE2A (0.43)
SCHEMBL7850567 0.69 PDE2A (0.43)
SCHEMBL7408950 0.69
SCHEMBL1388119 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708774-B1 IMIDAZO[1,2-a]PYRAZIN-4-ONE DERIVATIVES ANTAGONISTS OF AMPA AND NMDA RECEPTORS RHONE POULENC RORER SA (FR) 1999-03-17 EP disclosed
EP-0708774-A1 IMIDAZO [1,2-A]PYRAZINE-4-ONE, PREPARATION THEREOF AND DRUGS CONTAINING SAME Aventis Pharma S.A. (FR) 1996-05-01 EP disclosed
WO-1995002601-A1 IMIDAZO[1,2-a]PYRAZINE-4-ONE, PREPARATION THEREOF AND DRUGS CONTAINING SAME RHONE-POULENC RORER S.A. (FR) 1995-01-26 WO disclosed