SCHEMBL8315812

SCHEMBL8315812

COc1ccc(/C=C/c2nc3c(s2)NCCCC3)cc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 2/20 0.43
RECQL P46063 1/20 0.40
KMT2A Q03164 6/20 0.39
MEN1 O00255 5/20 0.39
NPC1 O15118 1/20 0.39
POLB P06746 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 4/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPK1 P28482 1/20 0.36
CTSL P07711 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
HPGD P15428 2/20 0.35
APP P05067 2/20 0.35
MAPT P10636 2/20 0.34
GFER P55789 1/20 0.34
LMNA P02545 1/20 0.34
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315815 1.00 TUBB1 (0.43) TUBB1RECQLKMT2AMEN1NPC1
SCHEMBL9694219 0.90 ALDH1A1 (0.45) TUBB1ALDH1A1SMN1; SMN2CYP1A2HPGD
SCHEMBL9694216 0.90 ALDH1A1 (0.45) TUBB1ALDH1A1SMN1; SMN2CYP1A2HPGD
Hydrochloric Acid SCHEMBL8316467 0.89 ALDH1A1 (0.44) TUBB1ALDH1A1SMN1; SMN2CYP1A2HPGD
Hydrochloric Acid SCHEMBL8316464 0.89 ALDH1A1 (0.44) TUBB1ALDH1A1SMN1; SMN2CYP1A2HPGD
SCHEMBL8313688 0.88 TUBB1 (0.36) TUBB1KMT2AMEN1NPC1POLB
SCHEMBL8313691 0.88 TUBB1 (0.36) TUBB1KMT2AMEN1NPC1POLB
SCHEMBL8315945 0.87 APP (0.45) TUBB1KMT2AMEN1ALDH1A1APP
SCHEMBL8315946 0.87 APP (0.45) TUBB1KMT2AMEN1ALDH1A1APP
Hydrochloric Acid SCHEMBL8317323 0.86 APP (0.44) TUBB1KMT2AMEN1ALDH1A1APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0351856-B1 Thiazolo[5,4-b]azepine compounds TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-09-15 EP disclosed
US-4956360-A LIPOPEROXIDE INHIBITORS, ENZYME INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-09-11 US disclosed