SCHEMBL8315964

SCHEMBL8315964

CCONC(=O)COCCCCC(=O)N1CCc2c([nH]c3ccccc23)C1

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.65
HDAC1 Q13547 2/20 0.65
GPX4 P36969 1/20 0.54
TAAR1 Q96RJ0 1/20 0.51
TRPV1 Q8NER1 13/20 0.51
FAAH O00519 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13627286 0.90 HDAC6 (0.76) HDAC6HDAC1GPX4TAAR1TRPV1
SCHEMBL5775992 0.89 HDAC6 (0.78) HDAC6HDAC1GPX4TAAR1TRPV1
SCHEMBL8315949 0.87 HDAC6 (0.61) HDAC6HDAC1GPX4TAAR1TRPV1
SCHEMBL8324393 0.86 HDAC6 (0.59) HDAC6HDAC1GPX4TAAR1TRPV1
SCHEMBL18688569 0.81 HDAC6 (0.77) HDAC6HDAC1GPX4TAAR1TRPV1
SCHEMBL8252701 0.79 HDAC6 (1.00) HDAC6HDAC1GPX4TAAR1TRPV1
SCHEMBL8320157 0.77 HDAC6 (0.74) HDAC6HDAC1GPX4TAAR1TRPV1
SCHEMBL14924871 0.76 HDAC1 (0.54) HDAC6HDAC1GPX4TAAR1TRPV1
SCHEMBL12660615 0.76 TRPV1 (0.55) HDAC6HDAC1GPX4TAAR1TRPV1
SCHEMBL20882095 0.76 GPX4 (0.77) HDAC6HDAC1GPX4TRPV1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004113336-A1 CARBOLINE AND BETACARBOLINE DERIVATIVES FOR USE AS HDAC ENZYME INHIBITORS CHROMA THERAPEUTICS LIMITED (GB) 2004-12-29 WO disclosed