SCHEMBL8316653

SCHEMBL8316653

Nc1ccc2c(c1)C(=O)c1c-2[nH]c(=O)c2nccn12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIA1 P42261 1/20 0.42
GRIA2 P42262 1/20 0.42
GRIA3 P42263 1/20 0.42
GRIA4 P48058 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
PDE2A O00408 1/20 0.42
PDE6D O43924 1/20 0.42
PDE8A O60658 1/20 0.42
PDE5A O76074 1/20 0.42
PDE9A O76083 1/20 0.42
PDE8B O95263 1/20 0.42
PDE6A P16499 1/20 0.42
PDE6G P18545 1/20 0.42
PDE4A P27815 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314487 0.82 PDE2A (0.50) PDE2APDE6DPDE8APDE5APDE9A
SCHEMBL7415664 0.76
SCHEMBL7411619 0.75
SCHEMBL1387892 0.73 PDE2A (0.49) PDE2APDE6DPDE8APDE5APDE9A
SCHEMBL1387425 0.72 PDE2A (0.48) PDE2APDE6DPDE8APDE5APDE9A
SCHEMBL8315788 0.70
SCHEMBL8315791 0.70
SCHEMBL7845909 0.69 PDE2A (0.45) PDE2APDE6DPDE8APDE5APDE9A
SCHEMBL7845913 0.69 PDE2A (0.45) PDE2APDE6DPDE8APDE5APDE9A
SCHEMBL8801240 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0752991-B1 IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZIN-4-ONES ANTAGONISTS OF AMPA AND NMDA RECEPTORS RHONE POULENC RORER SA (FR) 1999-05-26 EP disclosed
EP-0752991-A1 INDENO[1,2-e]PYRAZINE-4-ONES, PREPARATION THEREOF AND DRUGS CONTAINING SAME Aventis Pharma S.A. (FR) 1997-01-15 EP disclosed
WO-1995026349-A1 INDENO[1,2-e]PYRAZINE-4-ONES, PREPARATION THEREOF AND DRUGS CONTAINING SAME RHONE-POULENC RORER S.A. (FR) 1995-10-05 WO disclosed