SCHEMBL8316697

SCHEMBL8316697

COC(=O)N1CCC(Nc2ncc3ncnc(Nc4cccc(C)c4)c3n2)CC1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.58
ERBB2 P04626 1/20 0.53
HPGD P15428 1/20 0.53
HTT P42858 1/20 0.53
IRAK4 Q9NWZ3 2/20 0.51
BRAF P15056 4/20 0.49
TYRO3 Q06418 1/20 0.47
MERTK Q12866 1/20 0.47
SYK P43405 2/20 0.47
KCNH2 Q12809 2/20 0.47
MAPK3 P27361 1/20 0.46
MAPK1 P28482 1/20 0.46
AURKB Q96GD4 1/20 0.46
GPR119 Q8TDV5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313532 0.93 EGFR (0.56) EGFRERBB2HPGDHTTBRAF
SCHEMBL8315160 0.91 EGFR (0.60) EGFRERBB2HPGDHTTBRAF
SCHEMBL8313473 0.90 EGFR (0.59) EGFRERBB2HPGDHTTBRAF
SCHEMBL8318765 0.90 EGFR (0.61) EGFRERBB2HPGDHTTBRAF
SCHEMBL6987353 0.89 EGFR (0.57) EGFRERBB2HPGDHTTBRAF
SCHEMBL7588633 0.87 EGFR (0.55) EGFRERBB2HPGDHTTBRAF
SCHEMBL7576084 0.87 EGFR (0.55) EGFRERBB2HPGDHTTBRAF
SCHEMBL8315128 0.86 EGFR (0.69) EGFRERBB2HPGDHTTBRAF
SCHEMBL8319428 0.86 EGFR (0.73) EGFRERBB2HPGDHTTBRAF
SCHEMBL7576095 0.86 EGFR (0.57) EGFRERBB2HPGDHTTBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed