SCHEMBL8317247

SCHEMBL8317247

CCCCc1ccc(C(=O)C2CCN(c3nc4ccc(S(=O)(=O)C5(CNO)CCOCC5)cc4s3)CC2)s1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.42
SMN1; SMN2 Q16637 6/20 0.42
RAB9A P51151 4/20 0.41
NPC1 O15118 3/20 0.41
TP53 P04637 9/20 0.41
ALDH1A1 P00352 3/20 0.40
LMNA P02545 3/20 0.40
STAT3 P40763 1/20 0.38
HTT P42858 1/20 0.38
GAA P10253 2/20 0.37
CYP2C9 P11712 2/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CTSK P43235 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312493 0.89 MMP13 (0.47) MAPTSMN1; SMN2TP53
Hydrochloric Acid SCHEMBL6264619 0.88 MMP13 (0.46) MAPTSMN1; SMN2TP53
SCHEMBL6234098 0.88 TP53 (0.44) MAPTSMN1; SMN2RAB9ANPC1TP53
SCHEMBL6286779 0.84 MAPT (0.40) MAPTSMN1; SMN2RAB9ANPC1TP53
SCHEMBL6229683 0.81 NPC1 (0.39) MAPTSMN1; SMN2RAB9ANPC1TP53
SCHEMBL8317378 0.72 MMP13 (0.52)
Hydrochloric Acid SCHEMBL6232519 0.71 MMP13 (0.51)
SCHEMBL6263388 0.70 MMP13 (0.41)
SCHEMBL8316792 0.69 MMP13 (0.43)
SCHEMBL6232760 0.67 MMP13 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048368-A2 HETEROARYLSULFONYLMETHYL HYDROXAMIC ACIDS AND AMIDES AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2004-06-10 WO disclosed