SCHEMBL8317769

SCHEMBL8317769

Cc1cccc(Nc2ncnc3cnc(N(C)C)nc23)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 1.00
HTT P42858 1/20 0.53
HIF1A Q16665 1/20 0.53
MAPK1 P28482 1/20 0.51
ERBB2 P04626 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314812 0.89 EGFR (0.79) EGFRHTTHIF1AMAPK1
SCHEMBL8316000 0.89 EGFR (0.79) EGFRHTTHIF1AMAPK1
SCHEMBL8318599 0.89 EGFR (0.79) EGFRHTTHIF1AMAPK1
SCHEMBL8319624 0.88 EGFR (0.78) EGFRHTTHIF1AMAPK1
SCHEMBL8318687 0.87 EGFR (0.77) EGFRHTTHIF1AMAPK1ERBB2
SCHEMBL8316168 0.85 EGFR (1.00) EGFRHTTHIF1AMAPK1ERBB2
SCHEMBL8316955 0.84 EGFR (0.72) EGFRHTTHIF1A
SCHEMBL8316963 0.84 EGFR (0.86) EGFRHTTHIF1AMAPK1ERBB2
SCHEMBL8318926 0.83 EGFR (0.71) EGFRHTTHIF1AMAPK1ERBB2
SCHEMBL8315552 0.82 EGFR (0.73) EGFRHTTHIF1AMAPK1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed