SCHEMBL8318422

SCHEMBL8318422

CCCn1c(=O)c2sc3nsnc3sc=2c1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 2/20 0.36
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PDE4A P27815 9/20 0.34
ADORA2A P29274 9/20 0.34
PDE4B Q07343 9/20 0.34
PDE4C Q08493 9/20 0.34
PDE4D Q08499 9/20 0.34
ADORA2B P29275 6/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 1/20 0.34
BLM P54132 1/20 0.34
PMP22 Q01453 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SIRT1 Q96EB6 1/20 0.32
SIRT3 Q9NTG7 1/20 0.32
SIRT5 Q9NXA8 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318449 0.86 TNF (0.52) TNFALDH1A1SMN1; SMN2ADORA2BCYP3A4
SCHEMBL8316287 0.84 GSK3B (0.32) TNFALDH1A1ADORA2BHSD17B10GSK3A
SCHEMBL23348857 0.67 L3MBTL1 (0.40) SMN1; SMN2PDE4AADORA2APDE4BPDE4C
SCHEMBL4307720 0.65 GSK3B (0.39) ALDH1A1ADORA2BCYP1A2HSD17B10GSK3A
SCHEMBL331903 0.61 PDE4A (0.47) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL6076720 0.58 TDP1 (0.52) ALDH1A1PDE4AADORA2APDE4BPDE4C
SCHEMBL8314445 0.58
SCHEMBL13232332 0.58
SCHEMBL4620773 0.57 GSK3B (0.38) ALDH1A1SMN1; SMN2PDE4AADORA2APDE4B
SCHEMBL1074421 0.57 L3MBTL1 (0.46) TNFALDH1A1SMN1; SMN2ADORA2BCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912580-A2 5H-PYRROLO(3',4':5,6)(1,4)DITHIINO(2,3-C)-(1,2,5)THIADIAZOLE-5,7(6H)-DIONE, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIAL AND MARINE ANTIFOULING AGENTS THE DOW CHEMICAL COMPANY (US) 1999-05-06 EP claimed
WO-1998001452-A2 5H-PYRROLO(3',4':5,6)(1,4)DITHIINO(2,3-C)-(1,2,5)THIADIAZOLE-5,7(6H)-DIONE, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIAL AND MARINE ANTIFOULING AGENTS THE DOW CHEMICAL COMPANY (US) 1998-01-15 WO claimed
US-5633219-A 5H-pyrrolo(3',4':5,6)(1,4)dithiino(2,3-C)(1,2,5)thiadiazole-5,7(6H)-dione, compositions containing them and their use as antimicrobial and marine antifouling agents THE DOW CHEMICAL COMPANY (US) 1997-05-27 US claimed
EP-0912580-A2 5H-PYRROLO(3',4':5,6)(1,4)DITHIINO(2,3-C)-(1,2,5)THIADIAZOLE-5,7(6H)-DIONE, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIAL AND MARINE ANTIFOULING AGENTS THE DOW CHEMICAL COMPANY (US) 1999-05-06 EP disclosed
WO-1998001452-A2 5H-PYRROLO(3',4':5,6)(1,4)DITHIINO(2,3-C)-(1,2,5)THIADIAZOLE-5,7(6H)-DIONE, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIAL AND MARINE ANTIFOULING AGENTS THE DOW CHEMICAL COMPANY (US) 1998-01-15 WO disclosed
US-5633219-A 5H-pyrrolo(3',4':5,6)(1,4)dithiino(2,3-C)(1,2,5)thiadiazole-5,7(6H)-dione, compositions containing them and their use as antimicrobial and marine antifouling agents THE DOW CHEMICAL COMPANY (US) 1997-05-27 US disclosed