SCHEMBL8319040

SCHEMBL8319040

CNC(=O)CCCNc1ncc2ncnc(Nc3ccc(F)c(Cl)c3)c2n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.54
ERBB2 P04626 13/20 0.54
HPGD P15428 1/20 0.54
HTT P42858 1/20 0.54
CSNK2A1 P68400 2/20 0.49
HDAC3 O15379 10/20 0.48
HDAC4 P56524 10/20 0.48
HDAC1 Q13547 10/20 0.48
HDAC7 Q8WUI4 10/20 0.48
HDAC2 Q92769 10/20 0.48
HDAC10 Q969S8 10/20 0.48
HDAC11 Q96DB2 10/20 0.48
HDAC8 Q9BY41 10/20 0.48
HDAC6 Q9UBN7 10/20 0.48
HDAC9 Q9UKV0 10/20 0.48
HDAC5 Q9UQL6 10/20 0.48
KDR P35968 1/20 0.47
MAPT P10636 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8317514 0.90 EGFR (0.54) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8319127 0.90 EGFR (0.54) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8314458 0.89 EGFR (0.53) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL6995363 0.87 EGFR (0.55) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8315925 0.85 EGFR (0.55) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL6994345 0.85 EGFR (0.53) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL6989432 0.85 STK17A (0.62) EGFRERBB2HPGDHTTMAPT
SCHEMBL8317956 0.85 EGFR (0.56) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL6990324 0.84 STK17A (0.59) EGFRERBB2HPGDHTTMAPT
SCHEMBL6999279 0.84 EGFR (0.56) EGFRERBB2HPGDHTTCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed