SCHEMBL8319663

SCHEMBL8319663

c1ccc(Oc2cccc3c2CCNC3)cc1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CD44 P16070 2/20 0.53
PNMT P11086 2/20 0.48
MAOB P27338 1/20 0.48
PRCP P42785 1/20 0.45
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
HTR1A P08908 4/20 0.44
SLC6A2 P23975 4/20 0.44
SLC6A4 P31645 4/20 0.44
SLC6A3 Q01959 4/20 0.44
P2RY1 P47900 1/20 0.41
HTR6 P50406 1/20 0.41
CARM1 Q86X55 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30519153 0.84 P2RY1 (0.48) CD44PNMTMAOBP2RY1
SCHEMBL25431215 0.84 P2RY1 (0.48) CD44PNMTMAOBP2RY1
Hydrochloric Acid SCHEMBL30519078 0.83 P2RY1 (0.47) CD44PNMTMAOBP2RY1
Hydrochloric Acid SCHEMBL25341340 0.83 P2RY1 (0.47) CD44PNMTMAOBP2RY1
SCHEMBL31233660 0.79 PNMT (0.56) CD44PNMTMAOBHTR2CHTR2B
SCHEMBL2358135 0.79 PNMT (0.56) CD44PNMTMAOBHTR2CHTR2B
Bromide SCHEMBL9719839 0.79 CARM1 (0.44) HTR2CHTR2BHTR1ASLC6A2SLC6A4
SCHEMBL5016341 0.78 RXRB (0.48) CD44HTR2CHTR2BHTR1ASLC6A2
Hydrochloric Acid SCHEMBL33527957 0.78 PNMT (0.55) CD44PNMTMAOBHTR2CHTR2B
Hydrochloric Acid SCHEMBL1124611 0.78 PNMT (0.55) CD44PNMTMAOBHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0687267-B1 PYRROLO-PYRIDINE DERIVATIVES AS LIGANDS OF DOPAMINE RECEPTOR MERCK SHARP & DOHME (GB) 1999-09-01 EP disclosed
US-5700809-A Pyrrolo-pyridine derivatives MERCK SHARP & DOHME, LTD. (GB) 1997-12-23 US disclosed
WO-1994020459-A2 PYRROLO-PYRIDINE DERIVATIVES AS DOPAMINE RECEPTOR LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1994-09-15 WO disclosed