SCHEMBL8320016

SCHEMBL8320016

COc1ccc(NCOc2ccc(NC(=O)C(F)(F)F)c(Br)c2)c(Br)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.45
TSHR P16473 1/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
POLB P06746 2/20 0.44
ALDH1A1 P00352 4/20 0.41
GAA P10253 2/20 0.41
THRB P10828 1/20 0.41
RXFP1 Q9HBX9 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MTNR1A P48039 4/20 0.41
MTNR1B P49286 4/20 0.41
NQO2 P16083 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
MAPT P10636 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29679686 0.88 NPSR1 (0.55) NPSR1TSHRMEN1KMT2APOLB
SCHEMBL5788197 0.88 NPSR1 (0.55) NPSR1TSHRMEN1KMT2APOLB
SCHEMBL8320012 0.81 NPSR1 (0.48) NPSR1TSHRMEN1KMT2APOLB
SCHEMBL27430704 0.74 TSHR (0.55) NPSR1TSHRMEN1KMT2AALDH1A1
SCHEMBL2552734 0.74 TSHR (0.74) NPSR1TSHRMEN1KMT2AALDH1A1
SCHEMBL29785065 0.74 TSHR (0.74) NPSR1TSHRMEN1KMT2AALDH1A1
SCHEMBL14409902 0.72 GAA (0.51) NPSR1TSHRMEN1KMT2AGAA
SCHEMBL7308049 0.72 TSHR (0.51) NPSR1TSHRMEN1KMT2AALDH1A1
SCHEMBL27010697 0.71 RAB9A (0.55) MEN1KMT2APOLBALDH1A1GAA
SCHEMBL15072456 0.71 NPC1 (0.47) MEN1KMT2APOLBALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929554-A1 SPIRO-AZACYCLIC DERIVATIVES, THEIR PREPARATION AND THEIR USE AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 1999-07-21 EP disclosed
WO-1998013369-A1 SPIRO-AZACYCLIC DERIVATIVES, THEIR PREPARATION AND THEIR USE AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1998-04-02 WO disclosed