SCHEMBL8320205

SCHEMBL8320205

CCCOc1ccc(CN(C)C2CCN(C)CC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.54
HTR2C P28335 2/20 0.54
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
LTA4H P09960 1/20 0.47
NOS2 P35228 1/20 0.47
HRH3 Q9Y5N1 2/20 0.45
NPC1 O15118 1/20 0.45
TP53 P04637 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
PRMT5 O14744 1/20 0.43
WDR77 Q9BQA1 1/20 0.43
HRH4 Q9H3N8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17285888 0.95 HTR2A (0.60) HTR2AHTR2CKDM4EALDH1A1LTA4H
SCHEMBL22878461 0.84 HTR2A (0.48) HTR2AHTR2CALDH1A1HRH3NPC1
SCHEMBL3569353 0.84 HRH3 (0.69) HRH3
SCHEMBL17284448 0.83 HTR2A (0.47) HTR2AHTR2CALDH1A1HRH3NPC1
SCHEMBL8251941 0.81 HTR2A (0.58) HTR2AHTR2CKDM4EALDH1A1LTA4H
SCHEMBL17282051 0.81 HTR2A (0.46) HTR2AHTR2CALDH1A1HRH3NPC1
SCHEMBL17285945 0.80 LTA4H (0.56) HTR2AKDM4EALDH1A1LTA4HNOS2
SCHEMBL17286035 0.80 HTR2A (0.56) HTR2AKDM4EALDH1A1LTA4HNOS2
SCHEMBL13887902 0.78 KDM4E (0.58) HTR2AHTR2CKDM4EALDH1A1LTA4H
SCHEMBL18412166 0.77 KDM4E (0.57) HTR2AHTR2CKDM4EALDH1A1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004066960-A2 COMBINATION OF H1, H3 AND H4 RECEPTOR ANTAGONISTS FOR TREATMENT OF ALLERGIC AND NON-ALLERGIC PULMONARY INFLAMMATION, CONGESTION AND ALLERGIC RHINITIS SCHERING CORPORATION (US) 2004-08-12 WO disclosed