SCHEMBL8320734

SCHEMBL8320734

O=C(O)CCOc1cccc2c1Cc1sc(S)nc1-2

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.44
LMNA P02545 1/20 0.41
FABP3 P05413 2/20 0.37
FABP4 P15090 2/20 0.37
S1PR5 Q9H228 7/20 0.35
ALDH1A1 P00352 2/20 0.35
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
FBP1 P09467 4/20 0.35
PDE10A Q9Y233 2/20 0.34
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7531034 0.94 ADORA1 (0.43) ADORA1FABP3FABP4S1PR5
SCHEMBL7521598 0.89 ADORA1 (0.45) ADORA1ALDH1A1CASP1SMN1; SMN2KDM4E
SCHEMBL7518668 0.85 ADORA1 (0.41) ADORA1ALDH1A1FBP1
SCHEMBL7520497 0.79 ADORA1 (0.40) ADORA1LMNAFABP3FABP4S1PR5
SCHEMBL7526025 0.79 KDM4E (0.42) ADORA1ALDH1A1CASP1SMN1; SMN2KDM4E
SCHEMBL7974210 0.77 ADORA1 (0.41) ADORA1LMNAFABP4TP53SMN1; SMN2
SCHEMBL7518636 0.77 ALDH1A1 (0.41) ADORA1LMNAALDH1A1KDM4EHPGD
SCHEMBL7522397 0.77 ADORA1 (0.38) ADORA1LMNAFABP3FABP4ALDH1A1
SCHEMBL7526545 0.75 ADORA1 (0.38) ADORA1FABP3FABP4S1PR5ALDH1A1
SCHEMBL7528838 0.74 ADORA1 (0.39) ADORA1FABP3FABP4S1PR5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929534-A1 TRYCYCLIC COMPOUNDS AS PROSTAGLANDIN I2 RECEPTOR AGONISTS Takeda Pharmaceutical Company Limited (JP) 1999-07-21 EP disclosed
WO-1998013356-A1 TRYCYCLIC COMPOUNDS AS PROSTAGLANDIN I2 RECEPTOR AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-04-02 WO disclosed