SCHEMBL8321986

SCHEMBL8321986

CC(N)(Cc1ccccc1)Cc1cccc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.48
TAAR1 Q96RJ0 1/20 0.48
CYP2D6 P10635 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
SIGMAR1 Q99720 3/20 0.42
NR1I2 O75469 1/20 0.42
LMNA P02545 1/20 0.42
ADRA2A P08913 1/20 0.42
ACHE P22303 1/20 0.42
HTR2A P28223 1/20 0.42
SLC6A4 P31645 1/20 0.42
KCNH2 Q12809 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CYP2C9 P11712 1/20 0.42
CASR P41180 1/20 0.41
MMP8 P22894 1/20 0.41
KMT2A Q03164 1/20 0.39
SSTR4 P31391 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL2412475 0.90 CYP1A2 (0.48) SLC6A2CYP2D6CYP1A2CYP2C19SIGMAR1
SCHEMBL30119619 0.83 CYP1A2 (0.46) SLC6A2CYP2D6CYP1A2CYP2C19SIGMAR1
SCHEMBL7037475 0.80 CYP1A2 (0.50) SLC6A2TAAR1CYP2D6CYP1A2CYP2C19
SCHEMBL516033 0.80 TAAR1 (0.73) SLC6A2TAAR1CYP2D6CYP1A2CYP2C19
Hydrochloric Acid SCHEMBL7217846 0.79 CYP1A2 (0.48) SLC6A2TAAR1CYP2D6CYP1A2CYP2C19
Ammonia Solution, Strong SCHEMBL2477835 0.78 SLC6A2 (0.70) SLC6A2TAAR1CYP2D6CYP1A2CYP2C19
SCHEMBL808870 0.77 TDP1 (0.53) SLC6A2CYP2D6CYP1A2CYP2C19SIGMAR1
SCHEMBL31675157 0.76 CYP2D6 (0.53) SLC6A2CYP2D6CYP1A2CYP2C19SIGMAR1
SCHEMBL11586023 0.76 CYP2D6 (0.53) SLC6A2CYP2D6CYP1A2CYP2C19SIGMAR1
SCHEMBL29981949 0.75 TDP1 (0.53) CYP1A2TDP1CASRKMT2ASSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed