SCHEMBL8322127

SCHEMBL8322127

C=C(O)CCCC(Nc1ncnc2cc(C(=O)N3CC=CC3)c(Cl)cc12)c1nc2cc(Cl)ccc2[nH]1

nearest known ligand 0.31

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.31
ITGAV P06756 1/20 0.31
ITGA5 P08648 1/20 0.31
ITGB6 P18564 1/20 0.31
EGFR P00533 4/20 0.31
ERBB2 P04626 3/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
CNR2 P34972 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30
CTDSP1 Q9GZU7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4154124 0.94 CNR1 (0.35) CNR1ITGAVITGA5ITGB6EGFR
SCHEMBL8317288 0.91 CNR1 (0.36) CNR1ITGAVITGA5ITGB6EGFR
SCHEMBL3003700 0.89 EGFR (0.35) EGFRERBB2ALDH1A1LMNAHRH4
SCHEMBL4162062 0.89 AURKA (0.33) CNR1ITGAVITGA5ITGB6EGFR
SCHEMBL4158304 0.88 EPHA2 (0.33) CNR1ITGAVITGA5ITGB6EGFR
SCHEMBL13772294 0.88 RPS6KB1 (0.33) CNR1ALDH1A1LMNAHRH4CNR2
SCHEMBL3000212 0.88 RPS6KB1 (0.33) CNR1ALDH1A1LMNAHRH4CNR2
SCHEMBL8320265 0.88 RPS6KB1 (0.33) CNR1ALDH1A1LMNAHRH4CNR2
SCHEMBL2992118 0.87 ALDH1A1 (0.44) ALDH1A1LMNA
SCHEMBL2995895 0.87 ITGAV (0.37) ITGAVITGA5ITGB6EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004058743-A1 NOVEL SUBSTITUTED NITROGEN-CONTAINING HETEROBICYCLES AND USE THEREOF AS FACTOR XA INHIBITORS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-07-15 WO disclosed