SCHEMBL8322963

SCHEMBL8322963

CCCCCCCCCCCCC(CC)C(=S)Nc1c(SC)cc(C)nc1SC

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SOAT1 P35610 6/20 0.34
LMNA P02545 1/20 0.30
GPR84 Q9NQS5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8321429 0.95 SOAT1 (0.35) SOAT1GPR84
SCHEMBL8324413 0.95 SOAT1 (0.35) SOAT1GPR84
SCHEMBL8319647 0.95 SOAT1 (0.35) SOAT1GPR84
SCHEMBL8325251 0.88 SOAT1 (0.34) SOAT1GPR84
SCHEMBL8323636 0.84 SOAT1 (0.38) SOAT1LMNA
SCHEMBL8322821 0.83
SCHEMBL9225520 0.82 SOAT1 (0.38) SOAT1
SCHEMBL9225723 0.79 SOAT1 (0.38) SOAT1GPR84
SCHEMBL8323297 0.78 LMNA (0.31) LMNA
SCHEMBL8323237 0.78 LMNA (0.31) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609960-B1 New N-heteroarylamide derivatives as inhibitors of acyl coenzyme A: cholestrol acyl transferase PFIZER (US) 1999-03-03 EP disclosed
US-5656634-A N-aryl and N-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme A: cholesterol acyl transferase (ACAT) PFIZER INC. (US) 1997-08-12 US disclosed
US-5362878-A Intermediates for making N-aryl and N-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme A: cholesterol acyl transferase (ACAT) PFIZER INC. (US) 1994-11-08 US disclosed
EP-0609960-A1 New N-heteroarylamide derivatives as inhibitors of acyl coenzyme A: cholestrol acyl transferase PFIZER INC. (US) 1994-08-10 EP disclosed