SCHEMBL8323191

SCHEMBL8323191

COC(=O)c1[nH]c2c(C)ccc(C)c2c1CN

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
LOXL2 Q9Y4K0 2/20 0.38
NR4A2 P43354 1/20 0.35
KDM4E B2RXH2 5/20 0.35
HPGD P15428 2/20 0.35
MAPK1 P28482 1/20 0.35
HTR6 P50406 1/20 0.34
ALDH1A1 P00352 3/20 0.34
HSD17B10 Q99714 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPT P10636 3/20 0.33
GAA P10253 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
HTT P42858 1/20 0.33
PADI4 Q9UM07 1/20 0.33
USP2 O75604 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322259 0.87 CYP1A2 (0.48) CYP1A2CYP3A4CYP2C19NR4A2KDM4E
SCHEMBL8318646 0.82 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C19NR4A2KDM4E
SCHEMBL8324039 0.82 MAPK1 (0.52) CYP1A2CYP3A4CYP2C19KDM4EHPGD
SCHEMBL8324009 0.82 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C19NR4A2KDM4E
SCHEMBL8318534 0.81 KDM4E (0.46) CYP1A2CYP3A4CYP2C19NR4A2KDM4E
SCHEMBL8324480 0.78 NR4A2 (0.41) CYP1A2CYP3A4CYP2C19NR4A2KDM4E
SCHEMBL8324886 0.77 CYP1A2 (0.40) CYP1A2CYP3A4CYP2C19NR4A2KDM4E
SCHEMBL8326080 0.77 CYP1A2 (0.40) CYP1A2CYP3A4CYP2C19NR4A2KDM4E
SCHEMBL8321899 0.77 CYP1A2 (0.40) CYP1A2CYP3A4CYP2C19NR4A2KDM4E
SCHEMBL8323510 0.77 HPGD (0.39) CYP1A2CYP3A4CYP2C19NR4A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866594-A Indole-2-carboxylate derivatives and fungicidal compositions for agricultural or horticultural use containing the derivatives as active component OTSUKA KAGAKU KABUSHIKI KAISHA (JP) 1999-02-02 US disclosed
EP-0791582-A1 INDOLE-2-CARBOXYLIC ESTER DERIVATIVES AND AGRICULTURAL AND HORTICULTURAL BACTERIOCIDES CONTAINING THE SAME AS THE ACTIVE INGREDIENT OTSUKA KAGAKU KABUSHIKI KAISHA (JP) 1997-08-27 EP disclosed