SCHEMBL8323489

SCHEMBL8323489

CS(=O)(=O)OCC1Cc2cc3ccccc3n2CC1COS(C)(=O)=O

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.36
HTR2C P28335 5/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
SIGMAR1 Q99720 11/20 0.34
NOTUM Q6P988 1/20 0.32
HTR1A P08908 1/20 0.31
NOD2 Q9HC29 1/20 0.31
NOD1 Q9Y239 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323495 1.00 HTR2A (0.36) HTR2AHTR2CCYP1A2CYP3A4CYP2D6
SCHEMBL8323502 1.00 HTR2A (0.36) HTR2AHTR2CCYP1A2CYP3A4CYP2D6
SCHEMBL8448934 0.79 HTR2A (0.40) HTR2AHTR2CSIGMAR1HTR1A
SCHEMBL1999141 0.79 HTR2A (0.40) HTR2AHTR2CSIGMAR1HTR1A
SCHEMBL8329799 0.73 HTR2A (0.42) HTR2AHTR2CSIGMAR1NOTUMHTR1A
SCHEMBL8329798 0.73 HTR2A (0.42) HTR2AHTR2CSIGMAR1NOTUMHTR1A
SCHEMBL8329794 0.73 HTR2A (0.42) HTR2AHTR2CSIGMAR1NOTUMHTR1A
SCHEMBL234225 0.69 HTR2A (0.43) HTR2AHTR2CSIGMAR1NOTUM
SCHEMBL18911725 0.69 HTR2A (0.46) HTR2AHTR2CSIGMAR1NOTUM
SCHEMBL8655471 0.68 DRD2 (0.38) HTR2AHTR2CSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed