SCHEMBL8324244

SCHEMBL8324244

CC(=O)C(=Cc1ccccc1F)C(=O)O

nearest known ligand 0.79

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.73
CYP3A4 P08684 1/20 0.73
CYP2C9 P11712 1/20 0.73
CYP2C19 P33261 1/20 0.73
HIF1A Q16665 1/20 0.73
KDM4E B2RXH2 1/20 0.44
TRPA1 O75762 1/20 0.44
NFE2L2 Q16236 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
KMT2A Q03164 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
AKR1C3 P42330 1/20 0.40
ERN1 O75460 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3402801 0.81 CYP1A2 (0.58) CYP1A2CYP3A4CYP2C9CYP2C19HIF1A
SCHEMBL149582 0.81 CYP1A2 (0.58) CYP1A2CYP3A4CYP2C9CYP2C19HIF1A
SCHEMBL7378695 0.81 CYP1A2 (0.63) CYP1A2CYP3A4CYP2C9CYP2C19HIF1A
SCHEMBL7378697 0.81 CYP1A2 (0.63) CYP1A2CYP3A4CYP2C9CYP2C19HIF1A
SCHEMBL9475914 0.80 CYP1A2 (0.49) CYP1A2CYP3A4CYP2C9CYP2C19HIF1A
SCHEMBL9475919 0.80 CYP1A2 (0.49) CYP1A2CYP3A4CYP2C9CYP2C19HIF1A
SCHEMBL9477455 0.79 CA1 (0.52) CYP1A2CYP3A4CYP2C9CYP2C19HIF1A
SCHEMBL9477461 0.79 CA1 (0.52) CYP1A2CYP3A4CYP2C9CYP2C19HIF1A
SCHEMBL7274765 0.78 NFKB1 (0.50) CYP1A2CYP3A4CYP2C9CYP2C19HIF1A
SCHEMBL7316254 0.78 NFKB1 (0.50) CYP1A2CYP3A4CYP2C9CYP2C19HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0866708-A4 DIHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMA CORP (US) 1999-05-06 EP disclosed
EP-0866708-A1 DIHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 1998-09-30 EP disclosed
WO-1997017969-A1 DIHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 1997-05-22 WO disclosed