SCHEMBL8324532

SCHEMBL8324532

O=S(=O)(NCc1cccs1)c1ccc(CBr)cc1

nearest known ligand 0.74

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.64
POLB P06746 3/20 0.64
TDP1 Q9NUW8 1/20 0.64
LMNA P02545 5/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
USP2 O75604 1/20 0.52
MAPT P10636 1/20 0.52
HTT P42858 1/20 0.52
MAPK1 P28482 1/20 0.51
KDM4E B2RXH2 2/20 0.50
PKM P14618 1/20 0.50
TSHR P16473 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.48
GAA P10253 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11887767 0.85 KMT2A (0.68) ALDH1A1POLBTDP1LMNAMEN1
SCHEMBL5343785 0.83 ALDH1A1 (0.66) ALDH1A1POLBTDP1LMNAMEN1
SCHEMBL1874186 0.83 ALDH1A1 (0.68) ALDH1A1POLBTDP1LMNAMEN1
SCHEMBL12793685 0.82 ALDH1A1 (0.72) ALDH1A1POLBTDP1LMNAMEN1
SCHEMBL28003774 0.82 ALDH1A1 (0.72) ALDH1A1POLBTDP1LMNAMEN1
SCHEMBL28113726 0.82 ALDH1A1 (0.68) ALDH1A1POLBTDP1LMNAMEN1
SCHEMBL14484120 0.81 ALDH1A1 (0.66) ALDH1A1POLBTDP1LMNAMEN1
SCHEMBL3562140 0.79 ALDH1A1 (0.64) ALDH1A1POLBTDP1LMNAMEN1
SCHEMBL13712056 0.79 ALDH1A1 (0.64) ALDH1A1POLBTDP1LMNAMEN1
SCHEMBL10288218 0.78 POLB (0.63) ALDH1A1POLBTDP1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635018-B1 4-(1H-2-METHYLIMIDAZO[4,5-c]PYRIDINYLMETHYL)PHENYLSULPHONAMIDE DERIVATIVES AS ANTAGONISTS OF PAF BRITISH BIO TECHNOLOGY (GB) 1999-12-22 EP disclosed
US-5516783-A PLATELET ACTIVATING FACTOR BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1996-05-14 US disclosed
EP-0635018-A1 4-(1H-2-METHYLIMIDAZO 4,5-c]PYRIDINYLMETHYL)PHENYLSULPHONAMIDE DERIVATIVES AS ANTAGONISTS OF PAF BRITISH BIO-TECHNOLOGY LIMITED (GB) 1995-01-25 EP disclosed
WO-1993016075-A1 4-(1H-2-METHYLIMIDAZO[4,5-c]PYRIDINYLMETHYL)PHENYLSULPHONAMIDE DERIVATIVES AS ANTAGONISTS OF PAF BRITISH BIO-TECHNOLOGY LIMITED (GB) 1993-08-19 WO disclosed