SCHEMBL8324762

SCHEMBL8324762

Clc1ccc2c(c1)CN(C1CCNCC1)Cc1nnc(C3CCN(c4ccccn4)CC3)n1-2

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 15/20 0.72
AVPR2 P30518 7/20 0.72
KCNH2 Q12809 4/20 0.72
OXTR P30559 3/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5101961 0.99 AVPR1A (0.71) AVPR1AAVPR2KCNH2OXTR
SCHEMBL5101634 0.95 AVPR1A (0.70) AVPR1AAVPR2KCNH2OXTR
SCHEMBL20727358 0.94 AVPR2 (0.79) AVPR1AAVPR2KCNH2OXTR
SCHEMBL20727315 0.93 OXTR (0.79) AVPR1AAVPR2KCNH2OXTR
SCHEMBL5101984 0.92 AVPR1A (0.73) AVPR1AAVPR2KCNH2OXTR
SCHEMBL5102057 0.90 AVPR1A (0.72) AVPR1AAVPR2KCNH2OXTR
SCHEMBL20727363 0.89 AVPR1A (0.73) AVPR1AAVPR2KCNH2OXTR
SCHEMBL5108491 0.88 AVPR1A (0.81) AVPR1AAVPR2KCNH2OXTR
SCHEMBL8322332 0.88 AVPR1A (0.64) AVPR1AAVPR2KCNH2OXTR
Hydrochloric Acid SCHEMBL5107857 0.87 AVPR1A (0.64) AVPR1AAVPR2KCNH2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7442795-B2 Triazole compounds useful in therapy PFIZER INC. (US) 2008-10-28 US disclosed
US-7442795-B2 Triazole compounds useful in therapy PFIZER INC. (US) 2008-10-28 US disclosed
WO-2004074291-A1 TRIAZOLE COMPOUNDS USEFUL IN THERAPY PFIZER LIMITED (GB) 2004-09-02 WO disclosed