SCHEMBL8325209

SCHEMBL8325209

CC(C)(C)OC(=O)/C=C/c1ccc(Cc2ncc(C3CCCCC3)[nH]2)cc1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 11/20 0.49
BRS3 P32247 1/20 0.41
CCR5 P51681 3/20 0.38
DGAT1 O75907 3/20 0.37
KDM1A O60341 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322805 0.84 BRS3 (0.48) NR1H4BRS3CCR5HDAC8HDAC6
SCHEMBL8321377 0.82 BRS3 (0.41) NR1H4BRS3CCR5HDAC8HDAC6
SCHEMBL8324028 0.80 NR1H4 (0.40) NR1H4BRS3KDM1AHDAC8HDAC6
SCHEMBL8325359 0.76 CA12 (0.43) NR1H4
SCHEMBL8319084 0.73 TAAR1 (0.43) NR1H4KDM1AHDAC8HDAC6
SCHEMBL8323886 0.73 NR1H4 (0.40) NR1H4BRS3HDAC8HDAC6
SCHEMBL8324344 0.73 HDAC8 (0.41) NR1H4KDM1AHDAC8HDAC6
SCHEMBL8325041 0.69 HDAC3 (0.42) NR1H4DGAT1HDAC8HDAC6
SCHEMBL8325020 0.69 NR1H4 (0.45) NR1H4HDAC8HDAC6
SCHEMBL19717163 0.69 HDAC8 (0.51) NR1H4KDM1AHDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed