SCHEMBL8324028

SCHEMBL8324028

CC(C)(C)OC(=O)/C=C/c1ccc(Cc2ncc(C(C)(C)C)[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 6/20 0.40
BRS3 P32247 1/20 0.40
ESR1 P03372 1/20 0.38
HDAC8 Q9BY41 3/20 0.37
HDAC6 Q9UBN7 2/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CA7 P43166 2/20 0.36
CA9 Q16790 2/20 0.36
CA14 Q9ULX7 2/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322760 0.86 TBXAS1 (0.48) BRS3ESR1HDAC8HDAC6HDAC3
SCHEMBL8323151 0.84 HDAC1 (0.54) HDAC8HDAC6HDAC3HDAC4HDAC1
SCHEMBL8325359 0.82 CA12 (0.43) NR1H4CA12CA1CA7CA9
SCHEMBL8325209 0.80 NR1H4 (0.49) NR1H4BRS3HDAC8HDAC6KDM1A
SCHEMBL8319084 0.79 TAAR1 (0.43) NR1H4ESR1HDAC8HDAC6HDAC3
SCHEMBL8323886 0.79 NR1H4 (0.40) NR1H4BRS3ESR1HDAC8HDAC6
SCHEMBL8324344 0.76 HDAC8 (0.41) NR1H4ESR1HDAC8HDAC6HDAC3
SCHEMBL8325041 0.75 HDAC3 (0.42) NR1H4HDAC8HDAC6HDAC3HDAC4
SCHEMBL19717163 0.74 HDAC8 (0.51) NR1H4ESR1HDAC8HDAC6HDAC2
SCHEMBL13845314 0.74 CA12 (0.53) NR1H4ESR1HDAC1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed