SCHEMBL8325585

SCHEMBL8325585

CCOC(=O)c1cnc2nc(OCC)cnc2c1Nc1ccc(OC)cc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 13/20 0.56
PDE4B Q07343 1/20 0.56
NPSR1 Q6W5P4 2/20 0.52
NPC1 O15118 1/20 0.51
TP53 P04637 4/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
THRB P10828 1/20 0.49
GAA P10253 2/20 0.47
MEN1 O00255 1/20 0.47
SLC2A1 P11166 1/20 0.47
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HTT P42858 1/20 0.47
CLK1 P49759 1/20 0.47
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8327776 0.98 MAPT (0.54) MAPTPDE4BNPSR1NPC1TP53
SCHEMBL8330781 0.90 GAA (0.47) MAPTPDE4BNPSR1NPC1SMN1; SMN2
SCHEMBL8561277 0.86 PDE4B (0.61) MAPTPDE4BNPSR1NPC1TP53
Hydrochloric Acid SCHEMBL8563873 0.85 PDE4B (0.60) MAPTPDE4BNPSR1NPC1TP53
SCHEMBL8325775 0.84 MAPT (0.56) MAPTPDE4BNPSR1NPC1TP53
Hydrochloric Acid SCHEMBL8330855 0.83 MAPT (0.56) MAPTPDE4BNPSR1NPC1TP53
Hydrochloric Acid SCHEMBL8330455 0.82 MAPT (0.55) MAPTPDE4BNPSR1NPC1TP53
SCHEMBL8328847 0.80 PDE4B (0.56) MAPTPDE4BNPSR1TP53SMN1; SMN2
SCHEMBL8563738 0.79 PDE4B (0.63) MAPTPDE4BNPSR1NPC1TP53
Hydrochloric Acid SCHEMBL8567124 0.78 PDE4B (0.62) MAPTPDE4BNPSR1NPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705260-B1 CONDENSED 4-AMINOPYRIDINES WITH ANTIRHEUMATIC ACTIVITY KNOLL AG (DE) 1999-03-03 EP claimed
EP-0705260-B1 CONDENSED 4-AMINOPYRIDINES WITH ANTIRHEUMATIC ACTIVITY KNOLL AG (DE) 1999-03-03 EP disclosed
US-5780482-A TREATING RHEUMATIC DISEASES KNOLL AKTIENGESELLSCHAFT (DE) 1998-07-14 US disclosed
WO-1995000511-A1 CONDENSED 4-AMINOPYRIDINES WITH ANTIRHEUMATIC ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed