SCHEMBL8326595

SCHEMBL8326595

CCOC(=O)CNCc1nc2ccccc2[nH]1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.70
MAPT P10636 3/20 0.67
ALDH1A1 P00352 5/20 0.61
LMNA P02545 2/20 0.61
RAB9A P51151 2/20 0.61
NPC1 O15118 1/20 0.61
MAPK1 P28482 1/20 0.61
SMN1; SMN2 Q16637 4/20 0.56
KDM4E B2RXH2 2/20 0.56
KMT2A Q03164 2/20 0.54
PKM P14618 2/20 0.52
DDAH1 O94760 1/20 0.50
HTT P42858 1/20 0.49
MYC P01106 1/20 0.48
TSHR P16473 1/20 0.48
MAPK10 P53779 1/20 0.48
GAA P10253 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12643754 0.86 HSD17B10 (0.65) HSD17B10MAPTALDH1A1LMNARAB9A
SCHEMBL7364475 0.85 GRIN2B (0.53) HSD17B10MAPTALDH1A1LMNARAB9A
SCHEMBL31529600 0.82 HSD17B10 (1.00) HSD17B10MAPTALDH1A1LMNARAB9A
SCHEMBL1218749 0.82 HSD17B10 (1.00) HSD17B10MAPTALDH1A1LMNARAB9A
SCHEMBL944969 0.80 MAPT (1.00) HSD17B10MAPTALDH1A1LMNARAB9A
SCHEMBL8443937 0.77 PKM (0.68) HSD17B10MAPTALDH1A1RAB9ANPC1
SCHEMBL5395748 0.77 MAPT (0.83) HSD17B10MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL711507 0.77 PKM (0.71) HSD17B10RAB9ANPC1SMN1; SMN2KMT2A
SCHEMBL31734838 0.77 PKM (0.71) HSD17B10RAB9ANPC1SMN1; SMN2KMT2A
SCHEMBL14578158 0.76 MAPT (0.81) HSD17B10MAPTALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed