SCHEMBL8327012

SCHEMBL8327012

c1cncc(-c2ncc3c(n2)-c2cccnc2CC3)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.46
DUSP10 Q9Y6W6 1/20 0.46
CYP11B1 P15538 5/20 0.41
CYP11B2 P19099 5/20 0.41
CYP19A1 P11511 2/20 0.41
CYP17A1 P05093 1/20 0.41
ALDH1A1 P00352 4/20 0.40
CYP3A4 P08684 3/20 0.40
CYP1A2 P05177 3/20 0.40
HSD17B10 Q99714 2/20 0.40
TSHR P16473 2/20 0.40
CYP2D6 P10635 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
LMNA P02545 3/20 0.40
KDM4E B2RXH2 2/20 0.40
MAPT P10636 2/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326151 0.87 CYP1A2 (0.41) CYP2A6CYP11B1CYP11B2CYP19A1CYP17A1
SCHEMBL8325078 0.84 DUSP10 (0.47) DUSP10ALDH1A1CYP3A4CYP1A2LMNA
SCHEMBL8327915 0.83 CYP2A6 (0.45) CYP2A6CYP11B1CYP11B2CYP19A1CYP17A1
SCHEMBL8330251 0.83 DUSP10 (0.45) DUSP10ALDH1A1CYP3A4CYP1A2CYP2D6
SCHEMBL8326575 0.79 CCNA2 (0.58) DUSP10ALDH1A1CYP3A4CYP1A2HSD17B10
SCHEMBL10670682 0.76 KDM4E (0.67) DUSP10ALDH1A1CYP3A4CYP1A2HSD17B10
SCHEMBL14172822 0.75 CCNA2 (0.46) CYP2A6CYP11B1CYP11B2ALDH1A1LMNA
SCHEMBL14172846 0.74 CYP11B1 (0.47) CYP2A6CYP11B1CYP11B2CYP19A1CYP17A1
SCHEMBL14172825 0.74 CYP11B1 (0.43) CYP2A6CYP11B1CYP11B2CYP19A1ALDH1A1
SCHEMBL429796 0.70 CYP2A6 (0.40) CYP2A6CYP11B1CYP11B2CYP19A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915879-A1 NOVEL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-05-19 EP claimed
WO-1998001449-A1 NOVEL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-01-15 WO claimed
EP-0915879-A1 NOVEL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-05-19 EP disclosed
WO-1998001449-A1 NOVEL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-01-15 WO disclosed