SCHEMBL8326575

SCHEMBL8326575

CSc1ncc2c(n1)CCc1cnc(-c3cccnc3)nc1-2

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 17/20 0.58
CDK2 P24941 17/20 0.58
CDK1 P06493 1/20 0.46
CDK7 P50613 1/20 0.46
CDK5 Q00535 1/20 0.46
DUSP10 Q9Y6W6 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8325285 0.85 CCNA2 (0.54) CCNA2CDK2CDK1CDK7CDK5
SCHEMBL8326420 0.81 CCNA2 (0.67) CCNA2CDK2CDK1CDK7CDK5
SCHEMBL8324679 0.81 CCNA2 (0.59) CCNA2CDK2CDK1CDK7CDK5
SCHEMBL8326151 0.80 CYP1A2 (0.41) CCNA2CDK2ALDH1A1CYP1A2CYP3A4
SCHEMBL8327012 0.79 CYP2A6 (0.46) CCNA2CDK2DUSP10ALDH1A1CYP1A2
SCHEMBL8327915 0.76 CYP2A6 (0.45) ALDH1A1CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL14172822 0.76 CCNA2 (0.46) CCNA2CDK2ALDH1A1
SCHEMBL7513198 0.68 KDM4E (0.59) CCNA2CDK2DUSP10ALDH1A1CYP1A2
SCHEMBL8325078 0.68 DUSP10 (0.47) CCNA2CDK2DUSP10ALDH1A1CYP1A2
SCHEMBL14172846 0.68 CYP11B1 (0.47) CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915879-A1 NOVEL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-05-19 EP disclosed
WO-1998001449-A1 NOVEL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-01-15 WO disclosed