SCHEMBL8327019

SCHEMBL8327019

COc1ncc2c(n1)CCCC2=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
TSHR P16473 2/20 0.49
GRM5 P41594 7/20 0.46
MAOB P27338 3/20 0.46
MAOA P21397 2/20 0.46
MAPT P10636 3/20 0.45
USP2 O75604 1/20 0.45
TP53 P04637 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
CA9 Q16790 1/20 0.42
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7908025 0.77 SMN1; SMN2 (0.56) SMN1; SMN2NPC1RAB9ATSHRGRM5
SCHEMBL23657063 0.75 GRM5 (0.59) SMN1; SMN2NPC1RAB9ATSHRGRM5
SCHEMBL18652499 0.74 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9ATSHRGRM5
SCHEMBL13482119 0.74 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9ATSHRGRM5
SCHEMBL418947 0.74 ALDH1A1 (0.54) SMN1; SMN2NPC1RAB9ATSHRGRM5
SCHEMBL29649329 0.74 ALDH1A1 (0.54) SMN1; SMN2NPC1RAB9ATSHRGRM5
SCHEMBL10271999 0.73 SMN1; SMN2 (0.49) SMN1; SMN2NPC1RAB9ATSHRGRM5
SCHEMBL22965056 0.73 CYP1A2 (0.36) TSHRMAPTUSP2ALDH1A1MEN1
SCHEMBL2491161 0.73 SMN1; SMN2 (0.63) SMN1; SMN2NPC1RAB9ATSHRGRM5
SCHEMBL10220388 0.73 SMN1; SMN2 (0.49) SMN1; SMN2NPC1RAB9ATSHRGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108484606-B Pyrimido [4,5-f ] quinazoline compound and application thereof 江南大学 2020-03-06 CN disclosed
EP-0915879-A1 NOVEL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-05-19 EP disclosed
WO-1998001449-A1 NOVEL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-01-15 WO disclosed