SCHEMBL8327640

SCHEMBL8327640

CC(C(=O)OC(C)(C)C)c1cc2cc(N)ccc2o1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 2/20 0.48
CA2 P00918 2/20 0.39
ALOX5 P09917 1/20 0.38
NPC1 O15118 1/20 0.36
APP P05067 1/20 0.35
KDM4E B2RXH2 2/20 0.35
GLA P06280 2/20 0.35
GAA P10253 2/20 0.35
MAPT P10636 2/20 0.35
HPGD P15428 2/20 0.35
NR1H2 P55055 1/20 0.34
TAS1R3 Q7RTX0 3/20 0.34
TAS1R1 Q7RTX1 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
CASP1 P29466 1/20 0.33
BRCA1 P38398 1/20 0.33
CASP7 P55210 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7796052 0.80 FLT3 (0.56) FLT3CA2ALOX5NPC1KDM4E
SCHEMBL3487931 0.77 FLT3 (0.61) FLT3CA2NPC1KDM4EGLA
SCHEMBL550740 0.71 APP (0.48) NPC1APPKDM4EMAPTNR1H2
SCHEMBL4424911 0.71 TP53 (0.41) CA2ALOX5KDM4EMAPTHPGD
SCHEMBL5796124 0.70 APP (0.47) CA2APPKDM4EMAPTHPGD
SCHEMBL12795483 0.68 FLT3 (0.51) FLT3CA2NPC1KDM4ERAB9A
SCHEMBL27511220 0.67 FLT3 (0.47) FLT3CA2NPC1TAS1R3TAS1R1
SCHEMBL3488095 0.66 FLT3 (0.73) FLT3CA2NPC1KDM4EGLA
SCHEMBL211674 0.66 FLT3 (0.67) FLT3CA2NPC1KDM4EGLA
SCHEMBL30493800 0.66 FLT3 (0.61) FLT3CA2KDM4EMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed