SCHEMBL8327760

SCHEMBL8327760

O=C1c2ccccc2C(=O)N1CC1CN(Cc2ccc(Cl)cc2)CCO1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 9/20 0.60
CYP1A2 P05177 2/20 0.60
CYP2C9 P11712 2/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C19 P33261 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2768622 0.91 DRD4 (0.60) DRD4CYP1A2CYP2C9CYP3A4CYP2D6
SCHEMBL1502135 0.91 DRD4 (0.60) DRD4CYP1A2CYP2C9CYP3A4CYP2D6
SCHEMBL2768626 0.91 DRD4 (0.60) DRD4CYP1A2CYP2C9CYP3A4CYP2D6
SCHEMBL4504836 0.90 DRD4 (0.60) DRD4CYP1A2CYP2C9CYP3A4CYP2D6
SCHEMBL4024060 0.90 DRD4 (0.60) DRD4CYP1A2CYP2C9CYP3A4CYP2D6
SCHEMBL6230220 0.89 DRD4 (0.61) DRD4CYP1A2CYP2C9CYP3A4CYP2D6
SCHEMBL8330129 0.77 CYP2D6 (0.49) CYP2D6
SCHEMBL6162301 0.76 DRD4 (0.67) DRD4CYP1A2CYP2C9CYP3A4CYP2D6
SCHEMBL6165547 0.76 DRD4 (0.67) DRD4CYP1A2CYP2C9CYP3A4CYP2D6
SCHEMBL6162866 0.76 DRD4 (0.67) DRD4CYP1A2CYP2C9CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed