SCHEMBL8328024

SCHEMBL8328024

c1ccc2c(c1)cc1n2CC2CNCC2C1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.46
HTR2C P28335 5/20 0.46
BPTF Q12830 1/20 0.41
CHRNA7 P36544 4/20 0.36
CHRNB2 P17787 3/20 0.36
CHRNB4 P30926 3/20 0.36
CHRNA3 P32297 3/20 0.36
CHRNA4 P43681 3/20 0.36
NOTUM Q6P988 1/20 0.35
SIGMAR1 Q99720 6/20 0.34
HTR1A P08908 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328027 1.00 HTR2A (0.46) HTR2AHTR2CBPTFCHRNA7CHRNB2
Hydrochloric Acid SCHEMBL8327629 0.98 HTR2A (0.45) HTR2AHTR2CBPTFCHRNA7CHRNB2
Hydrochloric Acid SCHEMBL8327632 0.98 HTR2A (0.45) HTR2AHTR2CBPTFCHRNA7CHRNB2
Hydrochloric Acid SCHEMBL8327635 0.98 HTR2A (0.45) HTR2AHTR2CBPTFCHRNA7CHRNB2
Formic Acid SCHEMBL8324928 0.92 HTR2A (0.43) HTR2AHTR2CBPTFCHRNA7CHRNB2
Formic Acid SCHEMBL8324934 0.92 HTR2A (0.43) HTR2AHTR2CBPTFCHRNA7CHRNB2
Formic Acid SCHEMBL8324932 0.92 HTR2A (0.43) HTR2AHTR2CBPTFCHRNA7CHRNB2
SCHEMBL8321466 0.74 CYP2D6 (0.41) HTR2AHTR2CSIGMAR1
SCHEMBL8321461 0.74 CYP2D6 (0.41) HTR2AHTR2CSIGMAR1
SCHEMBL18911725 0.73 HTR2A (0.46) HTR2AHTR2CNOTUMSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed