SCHEMBL8328246

SCHEMBL8328246

c1ccc2c(c1)cc1n2CC2(CC1)CO2

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.49
HTR2C P28335 5/20 0.49
NOTUM Q6P988 1/20 0.38
SIGMAR1 Q99720 7/20 0.33
F9 P00740 2/20 0.31
HTR1A P08908 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL233434 0.80 HTR2A (0.44) HTR2AHTR2CNOTUMSIGMAR1
SCHEMBL18202247 0.78 HTR2A (0.47) HTR2AHTR2CNOTUMSIGMAR1HTR1A
SCHEMBL19921285 0.78 HTR2A (0.47) HTR2AHTR2CNOTUMSIGMAR1F9
SCHEMBL8322785 0.73 HTR2A (0.47) HTR2AHTR2CNOTUMSIGMAR1HTR1A
SCHEMBL8328872 0.73 HTR2A (0.47) HTR2AHTR2CNOTUMSIGMAR1HTR1A
SCHEMBL8328030 0.71 HTR2A (0.39) HTR2AHTR2CNOTUMSIGMAR1F9
SCHEMBL8328457 0.71 HTR2A (0.55) HTR2AHTR2CNOTUMSIGMAR1
SCHEMBL18911621 0.70 HTR2A (0.73) HTR2AHTR2CNOTUMSIGMAR1HTR1A
SCHEMBL9394920 0.69 HTR2A (0.43) HTR2AHTR2CNOTUM
SCHEMBL21028327 0.68 HTR2A (0.42) HTR2AHTR2CNOTUMSIGMAR1F9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed