SCHEMBL8328872

SCHEMBL8328872

NC1CC12CCc1cc3ccccc3n1C2

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.47
HTR2C P28335 5/20 0.47
NOTUM Q6P988 1/20 0.36
SIGMAR1 Q99720 9/20 0.33
HTR1A P08908 1/20 0.32
KDM1A O60341 1/20 0.31
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322785 1.00 HTR2A (0.47) HTR2AHTR2CNOTUMSIGMAR1HTR1A
SCHEMBL8328030 0.80 HTR2A (0.39) HTR2AHTR2CNOTUMSIGMAR1
SCHEMBL8322544 0.78 HTR2A (0.40) HTR2AHTR2CNOTUMSIGMAR1HTR1A
SCHEMBL18202247 0.75 HTR2A (0.47) HTR2AHTR2CNOTUMSIGMAR1HTR1A
SCHEMBL19921285 0.75 HTR2A (0.47) HTR2AHTR2CNOTUMSIGMAR1HTR1A
SCHEMBL8328246 0.73 HTR2A (0.49) HTR2AHTR2CNOTUMSIGMAR1HTR1A
SCHEMBL233434 0.72 HTR2A (0.44) HTR2AHTR2CNOTUMSIGMAR1
SCHEMBL8325934 0.71 HTR2A (0.34) HTR2AHTR2CSIGMAR1KDM1AMAOB
SCHEMBL231854 0.69 HTR2A (0.51) HTR2AHTR2CNOTUMSIGMAR1
SCHEMBL21028327 0.69 HTR2A (0.42) HTR2AHTR2CNOTUMSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed