SCHEMBL8328517

SCHEMBL8328517

CNCc1nc2c(OC)ccc(OC)c2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.41
PDE4A P27815 4/20 0.40
PDE4B Q07343 4/20 0.40
PDE4C Q08493 4/20 0.40
PDE4D Q08499 4/20 0.40
NQO2 P16083 1/20 0.37
HTR7 P34969 1/20 0.36
PIM1 P11309 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1012169 0.82 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DNQO2
SCHEMBL2269491 0.81 ADORA1 (0.50) PKMPDE4APDE4BPDE4CPDE4D
SCHEMBL5062073 0.80 PDE4A (0.42) PKMPDE4APDE4BPDE4CPDE4D
Ammonia Solution, Strong SCHEMBL3664643 0.75 KDM4E (0.39) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL30096766 0.75 CSNK2A2 (0.49) PKMPDE4APDE4BPDE4CPDE4D
SCHEMBL2849211 0.74 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DNQO2
SCHEMBL2841387 0.73 L3MBTL4 (0.38) PDE4APDE4BPDE4CPDE4D
SCHEMBL2543790 0.73 L3MBTL4 (0.38) PDE4APDE4BPDE4CPDE4DPOLB
SCHEMBL2840584 0.72 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DHTR7
SCHEMBL2272231 0.72 PDE4A (0.49) PKMPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
CN-1209744-A Vitronectin receptor antagonists SMITHKLINE BEECHAM CORP (US) 1999-03-03 CN disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed