SCHEMBL8328678

SCHEMBL8328678

c1ccc2c(c1)cc1n2CC2(CCNC2)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.47
HTR2C P28335 5/20 0.47
CYP11B1 P15538 1/20 0.38
TSHR P16473 3/20 0.36
USP2 O75604 6/20 0.34
CYP2D6 P10635 6/20 0.34
CYP1A2 P05177 5/20 0.34
ALDH1A1 P00352 5/20 0.34
CYP3A4 P08684 4/20 0.34
HSD17B10 Q99714 3/20 0.34
TP53 P04637 2/20 0.34
MAPK1 P28482 2/20 0.34
CYP2C9 P11712 1/20 0.34
HIF1A Q16665 1/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC6A3 Q01959 2/20 0.34
HPGD P15428 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323016 0.87 HTR2A (0.52) HTR2AHTR2CCYP11B1TSHRUSP2
SCHEMBL8322232 0.80 HTR2A (0.50) HTR2AHTR2CCYP11B1TSHRUSP2
SCHEMBL8328958 0.74 HTR2A (0.49) HTR2AHTR2CTSHRCYP2D6CYP1A2
SCHEMBL8327428 0.66 HTR2A (0.40) HTR2AHTR2CNOTUM
SCHEMBL19921285 0.65 HTR2A (0.47) HTR2AHTR2CNOTUM
SCHEMBL18202247 0.65 HTR2A (0.47) HTR2AHTR2CNOTUM
SCHEMBL8328457 0.65 HTR2A (0.55) HTR2AHTR2CTSHRCYP2D6CYP1A2
SCHEMBL233434 0.65 HTR2A (0.44) HTR2AHTR2CTSHRALDH1A1MAPK1
SCHEMBL2356686 0.64 HTR2A (1.00) HTR2AHTR2CNOTUM
SCHEMBL2591145 0.64 HTR2C (0.73) HTR2AHTR2CNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed